Donepezil

WHAT IS IT?

Donepezil (Aricept) is a cholinesterase inhibitor that works to decrease the rate of acetylcholine breakdown. This ultimately increases levels of acetylcholine in the synaptic cleft.

WHEN DO WE USE IT?

Alzheimer diseasepatients with this condition often will try cholinesterase inhibitors like Donepezil to slow disease progression (these are first-line medications).

WHEN DO WE AVOID USING IT?

Known hypersensitivity to the medication.

HOW IS IT ADMINISTERED?

Administered orally

Source
Source
WHAT ARE THE SIDE EFFECTS/TOXICITY?

Symptoms of increased acetylcholine: nausea, diarrhea, insomnia, vomiting, muscle cramps

FURTHER READING

DynaMed

UpToDate

 

Page Updated: 08.14.2016